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Bumetanide


Bumetanide

3-(aminosulfonyl)-5-(butylamino)-
4-phenoxybenzoic acid
CAS number
28395-03-1
ATC code
C03CA02
Chemical formula CH20N2O5S
Molecular weight 364.42
Bioavailability almost complete
Metabolism hepatic
Elimination half-life 60-90 minutes
Excretion renal
Pregnancy category C (Australia)
Legal status S4 (Aust)
POM (UK)
Routes of administration oral

Bumetanide is a loop diuretic of the sulfamyl category. It is often used in patients in whom high doses of furosemide are ineffective. There is however no reason not to use bumetanide as a first choice drug. The main difference between the two substances is in bioavailability. Furosemide is incompletely absorbed in the intestine (40%), and there is substantial inter- and intraindividual differences in bioavailability (range 10-90%). Bumetanide is completely absorbed (80%), and the absorption is not altered when it is taken with food. It is said to be a more predictable diuretic, meaning that the predictable absorption is reflected in a more predictable effect.

Bumetanide is 40 times more potent than furosemide (for patients with normal renal function).

01-04-2007 01:16:19
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